Leuprorelin Acetate CAS NO.74381-53-6
TECHNICAL SPECIFICATIONS
| Item | Specification |
|---|---|
| Product Name | Leuprorelin Acetate |
| CAS NO. | 74381-53-6 |
| Appearance | White to off-white crystalline powder |
| Molecular Formula | C₅₉H₈₄N₁₆O₁₂S·C₂H₄O₂ |
| Molecular Weight | 1269.52 g/mol |
| Purity (RP-HPLC) | ≥98.0% |
| Solubility | Freely soluble in water, slightly soluble in methanol, practically insoluble in ether and chloroform. |
| Endotoxin | < 1.0 EU/mg |
| Biological Activity | Exhibits potent luteinizing hormone-releasing hormone (LHRH) agonist activity, suppressing gonadotropin secretion and reducing sex hormone levels. |
| Storage Conditions | Store at 2–8°C, protected from light and moisture. |
| Stock Location | Stock in USA |
| MOQ | 1g |
1.MECHANISM OF ACTION
Leuprorelin Acetate acts as a GnRH receptor agonist. Upon initial administration, it stimulates the pituitary gland to release LH and FSH, causing a temporary surge in sex hormone levels. With continuous administration, it downregulates GnRH receptors, leading to sustained suppression of LH and FSH secretion.
2.PRODUCT INDICATIONS
- Advanced Prostate Cancer: Palliative treatment in advanced or metastatic cases.
- Endometriosis: Management of pain and reduction of endometrial lesions.
- Central Precocious Puberty (CPP): For children with early onset of puberty.
- Uterine Fibroids: Preoperative management to reduce fibroid size and associated symptoms.
- Breast Cancer: Used in certain premenopausal hormone-receptor-positive cases.
3.CLINICAL EFFICACY OF PRODUCT
4.DELIVERY & SHIPPING
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Professional and Secure Packaging
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Shipping Methods
Main Method: International Air Freight
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